diazepam UK /dʌɪˈaz.ɪ.pam/US /daɪˈæz.əˌpæm/ noun1 •A tranquilizing muscle relaxant drug (trademark Valium) used mainly to relieve anxiety.2001: The most effective anti-anxiety drugs (tranquillizers) are the benzodiazepines, epitomized by diazepam (Valium®). — Leslie Iversen, Drugs: A Very Short Introduction (Oxford 2001, p. 57) — 2001 formsdiazepams